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KLHL12-In-7k | KLHL12-In-7k : Inhibitor of KLHL12
RATINGS:
Cellular Use: (0 reviews)

In Model Organisms: (0 reviews)
Probe Summary
Selectivity
Potency
In Vivo
Control Compounds
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Probe Summary

Targets Biochemical/Biophysical Potency Cellular Potency
KLHL12
  • Ki:330 nM
  • Kd:480 nM
  • IC50:140 nM
  • IC50:620 nM
Inhibitor
up to 1 uM

Selectivity

In Vitro Selectivity Assessment
Potency Assay Off-Target:
Selectivity was assessed computationally and based on sequence similarities within the family.
Selectivity Assessment Description:
Ten of KLHL family proteins share sequence identity above 35% and are thus considered highly homolog ...

Potency
Cellular
In Vitro

KLHL12

Mode of Action: Inhibitor

Structure-Activity-Relationship data available? Yes

DOI Reference: 10.1021/acs.jmedchem.5c02931

Chemical Information

Coming Soon...

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Expert Reviews

No SERP comments found for KLHL12-In-7k

Probe KLHL12-In-7k is in the process of SERP review.

Please continue to check back for new reviews and commentary.